@article{b60acef3655d45dea54f74973189e16e,
title = "Catalytic enantioselective synthesis of key intermediates for NET inhibitors using atropisomeric lactam chemistry",
abstract = "An atropisomeric lactam which was prepared with high enantioselectivity by catalytic asymmetric intramolecular N-arylation, was efficiently converted to synthetic intermediates for NET inhibitors through highly diastereoselective α-alkylation followed by hydration and trans-tert-butylation.",
author = "Osamu Kitagawa and Daisuke Kurihara and Hajime Tanabe and Taichi Shibuya and Takeo Taguchi",
note = "Funding Information: We gratefully acknowledge Takasago International Corporation for supplying (R)-SEGPHOS. This work was partly supported by a Grant-in-Aid from The Research Foundation for Pharmaceutical Sciences, and a Grant-in-Aid [(C) Grant No. 18590018] for Scientific Research and the Ministry of Education, Science, Sports and Culture of Japan.",
year = "2008",
month = jan,
day = "14",
doi = "10.1016/j.tetlet.2007.11.101",
language = "English",
volume = "49",
pages = "471--474",
journal = "Tetrahedron Letters",
issn = "0040-4039",
publisher = "Elsevier Limited",
number = "3",
}